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uncompetitive, pore, mostly, putrescine, huperzine, diethylenetriamine, diaminopropane, 101676, arcaine, 9379, mrz, 576, 105519, 73068, 701324, 689560, harkoseride, 196771, gavestinel, 1328, cka, dcka, kyn, selfotel, 220581, ppda, perzinfotel, peaqx, pbpd, 17742, 12626, midafotel, cppene, 100453, 274614, 235959, 233053, cpp, 19755, 40116, 39551, 37849, ap7, ap5, apv, competitive, 718, plazinemdor, epipregnanolone, dehydroepiandrosterone, spermine, spermidine, neomycin, sarcosine, neboglamine, nebostinel, milacemide, 687, 414, 966, dimethylglycine, ccg, b6b21, acpc, acbd, tetrazolylglycine, quinolinic, homoquinolinic, homocysteic, hca, amaa, nmdar, 3763, 302, ns102, 382884, sym, 2081, 339434, kainic, atpa, iodowillardiine, bromowillardiine, kainate, kar, talampanel, rap, 219, perampanel, irampanel, 53655, 52466, zonampanel, ym90k, fanapanel, mpqx, becampanel, atpo, tulrampator, 47445, 1632, 18986, pramiracetam, piracetam, pesampator, biib, 104, 04958242, pepa, oxiracetam, 26576, 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85 ly 456 236 mcpg nps 2390 mglur 5 tooltip metabotropic glutamate receptor 5 agonists acpd adx 47273 cdppb chpg dfb dhpg glutamate ibotenic acid quisqualic acid vu 1545 positive allosteric modulators lsn2463359 antagonists ctep dmeob ly 344 545 mavoglurant mcpg nps 2390 remeglurant sib 1757 sib 1893 negative allosteric modulators azd9272 basimglurant dipraglurant fenobam grn 529 mpep mtep raseglurant zabaglurant group ii mglur 2 tooltip metabotropic glutamate receptor 2 agonists bina cbipes dcg iv eglumetad ly 354740 glutamate ibotenic acid ly 379 268 ly 487 379 ly 566 332 mgs 0028 pomaglumetad ly 404039 pomaglumetad methionil ly 2140023 talaglumetad ly 544344 positive allosteric modulators jnj 40411813 adx 71149 antagonists apica cecxg eglu hydia ly 307 452 ly 341 495 mcpg mgs 0039 pccg 4 negative allosteric modulators decoglurant ro4491533 mglur 3 tooltip metabotropic glutamate receptor 3 agonists cbipes dcg iv eglumetad ly 354740 glutamate ibotenic acid ly 379 268 ly 487 379 mgs 0028 pomaglumetad ly 404039 pomaglumetad methionil ly 2140023 talaglumetad ly 544344 antagonists apica cecxg eglu hydia ly 307 452 ly 341 495 mcpg mgs 0039 negative allosteric modulators decoglurant ro4491533 group iii mglur 4 tooltip metabotropic glutamate receptor 4 agonists glutamate l ap4 lsp2 9166 phccc vu 001 171 vu 0155 041 positive allosteric modulators foliglurax mpep antagonists cppg map4 mppg msop mtpg ubp 1112 mglur 6 tooltip metabotropic glutamate receptor 6 agonists glutamate l ap4 antagonists cppg map4 mppg msop mtpg ubp 1112 mglur 7 tooltip metabotropic glutamate receptor 7 agonists amn082 glutamate l ap4 lsp2 9166 antagonists cppg map4 mmpip mppg msop mtpg ubp 1112 xap044 negative allosteric modulators adx71743 mglur 8 tooltip metabotropic glutamate receptor 8 agonists dcpg glutamate l ap4 positive allosteric modulators az12216052 antagonists cppg map4 mppg msop mtpg ubp 1112 see also receptor signaling modulators ionotropic glutamate receptor modulators glutamate metabolism transport modulators v t e opioid receptor modulators μ opioid mor agonists abridged full list 3 ho pcp 7 acetoxymitragynine 7 hydroxymitragynine ψ akuammigine α chlornaltrexamine α narcotine acetyldihydrocodeine acetylfentanyl acrylfentanyl adrenorphin metorphamide ah 7921 akuammicine akuammidine alfentanil anileridine apparicine β endorphin bam 12p bam 18p bam 22p benzhydrocodone benzylmorphine bezitramide biphalin bu08070 buprenorphine butorphan butorphanol butyrfentanyl bw373u86 carfentanil casokefamide cebranopadol chloroxymorphamine codeine dadle damgo dago dermorphin desmetramadol desmethyltramadol desomorphine deumitragynine dextromoramide dextropropoxyphene propoxyphene dezocine dimenoxadol dimethylaminopivalophenone eluxadoline diamorphine heroin dihydrocodeine dihydroetorphine dihydromorphine dinalbuphine sebacate diphenoxylate dipipanone dynorphin a embutramide endomorphin 1 endomorphin 2 eseroline ethylmorphine etorphine fentanyl fluorophen frakefamide furanylfentanyl hemorphin 4 herkinorin hodgkinsine hydrocodone hydromorphinol hydromorphone ibntxa ketamine ketobemidone kratom laudanosine lefetamine leu enkephalin levacetylmethadol levomethorphan levorphanol lexanopadol loperamide loxicodegol ls 115509 matrine meb 1170 meptazinol met enkephalin metenkefalin methadone metkefamide metopon mitragynine mitragynine pseudoindoxyl morphiceptin morphine nalbuphine naloxone benzoylhydrazone nalbzoh nalmexone naltalimide neopine nfepp nicocodeine nicodicodine nicomorphine norketamine nufenoxole octreotide oliceridine oxycodegol nktr 181 oxymorphone 3 methoxynaltrexonazine om 3 mnz oripavine oxycodone oxymorphazone oxymorphonazine oxymorphone oxymorphone phenylhydrazone oxypnph papaver somniferum opium pentazocine pericine pethidine meperidine phenazocine phencyclidine piminodine piritramide pl 017 prodine propiram pzm21 racemethorphan racemorphan remifentanil salsolinol sc 17599 sinomenine sr 15099 sr 17018 sufentanil susineridine tapentadol tetrahydropapaveroline th 030418 thebaine thienorphine tianeptine tilidine tramadol trimebutine trimu 5 trv734 tubotaiwine u 47700 valorphin viminol xorphanol antagonists 3s 4s picenadol 2 s n n r viminol 3cs nalmefene 4 caffeoyl 1 5 quinide 4 hydroxyflavanone 4 7 dihydroxyflavone 6β naltrexol 6β naltrexol d4 18 mc α gliadin β chlornaltrexamine β funaltrexamine akuammine alvimopan am 251 apigenin at 076 axelopran bevenopran catechin catechin gallate clocinnamox ctap ctop cyclofoxy cyprodime diacetylnalorphine diprenorphine ecg egc epicatechin eptazocine gemazocine ginsenoside r hyperoside ibogaine jdtic levallorphan lobeline ly 255582 ly 2196044 methocinnamox methylnaltrexone methylsamidorphan naldemedine nalmefene nalodeine n allylnorcodeine nalorphine nalorphine dinicotinate naloxazone naloxegol naloxol naloxonazine naloxone naltrexazone naltrexonazine naltrexone naltrindole naringenin noribogaine oxilorphan pawhuskin a rimonabant quadazocine samidorphan taxifolin δ opioid dor agonists 3cs nalmefene 6 gnti 7 siom adl 5747 pf 04856881 adl 5859 alazocine skf 10047 amoxapine ar m100390 arm390 azd2327 β endorphin bam 18p biphalin bu 48 butorphan butorphanol bw373u86 casokefamide cebranopadol codeine cyclazocine dadle deltorphin a deltorphin i deltorphin ii desmethylclozapine desmetramadol desmethyltramadol dezocine diamorphine heroin dihydroetorphine dihydromorphine dpdpe dpi 221 dpi 3290 dslet ethylketazocine etorphine fentanyl fit fluorophen hemorphin 4 hydrocodone hydromorphone ibogaine isomethadone jnj 20788560 knt 127 kratom laudanosine leu enkephalin levomethorphan levorphanol lexanopadol lofentanil met enkephalin metenkefalin metazocine metkefamide mitragynine mitragynine pseudoindoxyl morphine n phenethyl 14 ethoxymetopon norbuprenorphine nalbzoh oripavine oxycodone oxymorphone pethidine meperidine proglumide racemethorphan racemorphan rwj 394674 samidorphan sb 235863 snc 80 snc 162 tan 67 sb 205 607 th 030418 thebaine thiobromadol c 8813 tonazocine tramadol trv250 xorphanol zenazocine antagonists 4 7 dihydroxyflavone 5 ntii 6β naltrexol 6β naltrexol d4 α santolol β chlornaltrexamine apigenin at 076 axelopran bevenopran bntx catechin catechin gallate clocinnamox diacetylnalorphine diprenorphine ecg egc eluxadoline epicatechin ici 154129 ici 174864 ly 255582 ly 2196044 methylnaltrexone methylnaltrindole n benzylnaltrindole nalmefene nalorphine naltrexone naltriben naltrindole naloxone naringenin noribogaine pawhuskin a quadazocine sdm25n sori 9409 taxifolin thienorphine κ opioid kor agonists 3cs nalmefene 4 allyl 6 oxa noribogainalog 6 gnti 8 cac 18 mc 14 methoxymetopon β chlornaltrexamine β funaltrexamine adrenorphin metorphamide akuammicine alazocine skf 10047 allomatrine apadoline asimadoline bam 12p bam 18p bam 22p big dynorphin bremazocine brl 52537 butorphan butorphanol bw373u86 cebranopadol ciprefadol cr665 cyclazocine cyclorphan cyprenorphine desmetramadol desmethyltramadol diamorphine heroin diacetylnalorphine difelikefalin dihydroetorphine dihydromorphine dinalbuphine sebacate diprenorphine dynorphin a dynorphin b rimorphin eluxadoline enadoline eptazocine erinacine e ethylketazocine etorphine fedotozine fentanyl gemazocine gr 89696 gr 103545 hemorphin 4 herkinorin hs665 hydromorphone hz 2 ibogaine ici 199 441 ici 204 448 ketamine ketazocine laudanosine leumorphin dynorphin b 29 levallorphan levomethorphan levorphanol lexanopadol lofentanil lpk 26 lufuradom matrine mb 1c oh meb 1170 menthol metazocine metkefamide mianserin mirtazapine morphine moxazocine mr 2034 n mppp nalbuphine nalbzoh nalfurafine nalmefene nalodeine n allylnorcodeine nalorphine naltriben niravoline norbuprenorphine norbuprenorphine 3 glucuronide noribogaine norketamine oripavine oxa noribogaine oxilorphan oxycodone pentazocine pethidine meperidine phenazocine proxorphan racemethorphan racemorphan rb 64 salvinorin a salvia salvinorin b ethoxymethyl ether salvinorin b methoxymethyl ether samidorphan spiradoline u 62066 th 030418 thienorphine tifluadom tricyclic antidepressants e g amitriptyline desipramine imipramine nortriptyline u 50488 u 54494a u 69593 xorphanol antagonists 4 hydroxyflavanone 4 7 dihydroxyflavone 5 gnti 6 gnti 6β naltrexol 6β naltrexol d4 β chlornaltrexamine buprenorphine samidorphan amentoflavone anti apigenin arodyne at 076 aticaprant axelopran az mtab binaltorphimine bu09059 buprenorphine catechin catechin gallate cerc 501 ly 2456302 clocinnamox cvl 354 cyclofoxy dezocine dippa egc ecg epicatechin hyperoside jdtic ly 255582 ly 2196044 ly 2444296 ly 2459989 ly 2795050 mejdtic methylnaltrexone ml190 ml350 mr 2266 n fluoropropyl jdtic naloxone naltrexone naltrindole naringenin navacaprant norbinaltorphimine noribogaine pawhuskin a pf 4455242 rb 64 ru 24213 quadazocine taxifolin uphit zyklophin nociceptin nop agonists arg14 lys15 nociceptin pf phe 4 nociceptin 1 13 nh 2 phe 1 ψ ch 2 nh gly 2 nociceptin 1 13 nh 2 ac ryyrwk nh 2 ac ryyrik nh 2 bu08070 buprenorphine cebranopadol dihydroetorphine etorphine jnj 19385899 levomethorphan levorphanol lexanopadol mcoppb mt 7716 nnc 63 0532 nociceptin orphanin fq nociceptin 1 11 nociceptin 1 13 nh 2 norbuprenorphine racemethorphan racemorphan ro64 6198 ro65 6570 sch 221510 sch 486757 sr 8993 sr 16435 sunobinop s 117957 th 030418 antagonists nphe 1 nociceptin 1 13 nh 2 at 076 ban orl 24 btrx 246040 ly 2940094 j 113397 jtc 801 nalbzoh nociceptin 1 7 nocistatin sb 612111 sr 16430 thienorphine trap 101 ufp 101 others enkephalinase inhibitors amastatin bl 2401 candoxatril d phenylalanine dexecadotril retorphan ecadotril sinorphan kelatorphan racecadotril acetorphan rb 101 rb 120 rb 3007 opiorphan selank semax spinorphin thiorphan tynorphin ubenimex bestatin propeptides β lipotropin proendorphin prodynorphin proenkephalin pronociceptin proopiomelanocortin pomc others kyotorphin met enkephalin releaser degradation stabilizer v t e progesterone receptor modulators pr tooltip progesterone receptor agonists progesterone derivatives 3β dihydroprogesterone 5α dihydroprogesterone 6α methylprogesterone 9α bromo 11 ketoprogesterone 11 dehydroprogesterone 11 deoxycorticosterone 16α hydroxyprogesterone 17α methyl 11 deoxycorticosterone acetate 20α dihydroprogesterone 20β dihydroprogesterone dimepregnen diosgenin p1 185 progesterone progesterone 3 acetyl enol ether quingestrone retroprogesterone derivatives 20α dihydrodydrogesterone 20α dihydrotrengestone du 41164 du 41165 dydrogesterone retroprogesterone ro 6 3129 trengestone 17α substituted progesterone derivatives 6α methyl 17α bromoprogesterone 15β hydroxycyproterone acetate 16 methylene 17α hydroxyprogesterone acetate 17α bromoprogesterone 17α hydroxyprogesterone hydroxyprogesterone 17α methylprogesterone acetomepregenol mepregenol diacetate algestone algestone acetonide algestone acetophenide anagestone anagestone acetate bromethenmadinone bromethenmadinone acetate butagest buterol chlormadinone chlormadinone acetate chlormadinone caproate chlormethenmadinone chlormethenmadinone acetate cismadinone cismadinone acetate clogestone clogestone acetate clomegestone clomegestone acetate cymegesolate cyproterone acetate delmadinone delmadinone acetate edogestrone flugestone flugestone acetate fluorometholone fluorometholone acetate flumedroxone flumedroxone acetate fluoromedroxyprogesterone acetate gestaclone gestobutanoyl haloprogesterone hydromadinone hydromadinone acetate hydroxyprogesterone acetate hydroxyprogesterone caproate hydroxyprogesterone hexanoate hydroxyprogesterone heptanoate hydroxyprogesterone enanthate hydroxyprogesterone heptanoate benzilic acid hydrazone mecigestone pentarane b medrogestone medroxyprogesterone medroxyprogesterone acetate medroxyprogesterone caproate megestrol megestrol acetate megestrol caproate melengestrol melengestrol acetate methenmadinone methenmadinone acetate methenmadinone caproate mometasone mometasone furoate osaterone osaterone acetate pentagestrone pentagestrone acetate pentarane a proligestone triamcinolone acetonide 19 norprogesterone derivatives 17α methyl 19 norprogesterone 18 methylsegesterone acetate 19 norprogesterone amadinone amadinone acetate demegestone fluoro ethyl norprogesterone fluoro furanyl norprogesterone gestadienol gestadienol acetate gestonorone acetate gestronol acetate gestonorone caproate gestronol hexanoate gestronol gestonorone nomegestrol nomegestrol acetate norgestomet org 2058 oxogestone oxogestone phenpropionate xinogestone promegestone segesterone segesterone acetate nestorone trimegestone testosterone derivatives progestins 6 6 difluoronorethisterone 6 6 difluoronorethisterone acetate 17α allyl 19 nortestosterone allylestrenol altrenogest chloroethynylnorgestrel cingestol danazol desogestrel dienogest ethinylandrostenediol ethandrostate ethisterone ethynerone etonogestrel etynodiol etynodiol diacetate gestodene gestrinone levonorgestrel levonorgestrel esters e g levonorgestrel butanoate lynestrenol lynestrenol phenylpropionate metynodiol metynodiol diacetate norelgestromin norethisterone norethindrone norethisterone esters e g norethisterone acetate norethisterone enanthate noretynodrel norgesterone norgestimate norgestrel norgestrienone norvinisterone oxendolone quingestanol quingestanol acetate tibolone tigestol tosagestin anabolic androgenic steroids 11β methyl 19 nortestosterone 11β methyl 19 nortestosterone dodecylcarbonate 19 nor 5 androstenediol 19 nor 5 androstenedione 19 nordehydroepiandrosterone bolandiol bolandiol dipropionate bolandione dimethisterone dienedione dienolone dimethandrolone dimethandrolone buciclate dimethandrolone dodecylcarbonate dimethandrolone undecanoate dimethyldienolone dimethyltrienolone ethyldienolone ethylestrenol ethylnandrol methyldienolone metribolone r 1881 methoxydienone methoxygonadiene mibolerone nandrolone nandrolone esters e g nandrolone decanoate nandrolone phenylpropionate norethandrolone normethandrone methylestrenolone normethandrolone normethisterone ru 2309 tetrahydrogestrinone trenbolone trienolone trenbolone esters e g trenbolone acetate trenbolone enanthate trendione trestolone trestolone acetate spirolactone derivatives canrenoic acid canrenone drospirenone mespirenone potassium canrenoate prorenone sc 5233 spirolactone sc 8109 spironolactone spirorenone nonsteroidal 3 8 dihydrodiligustilide lg 2527 lg 100128 riligustilide rwj 26819 rwj 49853 rwj 60130 tanaproget zm 182345 unknown org 47241 org 201745 mixed sprms tooltip selective progesterone receptor modulators steroidal dihydroethisterone 5α dihydrolevonorgestrel 5α dihydronorethisterone asoprisnil asoprisnil ecamate guggulsterone j1042 lg 120838 metapristone ru 42633 mifepristone ru 486 orf 9371 orf 9326 org 31710 org 33628 rmi 12936 telapristone ulipristal acetate vilaprisan zk 137316 nonsteroidal apigenin kaempferol lg 120920 naringenin pra 910 syringic acid antagonists steroidal aglepristone lilopristone lonaprisan onapristone org 31710 org 31806 org 33628 rti 3021 022 toripristone zanoterone nonsteroidal darolutamide lg 001447 lg 100127 lg 1...
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