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pressants amitriptyline butriptyline cianopramine clomipramine desipramine dosulepin dothiepin doxepin imipramine lofepramine melitracen nortriptyline protriptyline trimipramine tetracyclic antidepressants amoxapine maprotiline mianserin oxaprotiline setiptiline others amezinium metilsulfate antihistamines e g brompheniramine chlorphenamine pheniramine tripelennamine antipsychotics e g loxapine ziprasidone arylcyclohexylamines e g ketamine phencyclidine dopexamine ephenidine ginkgo biloba indeloxazine nefazodone opioids e g desmetramadol methadone pethidine meperidine tapentadol tramadol levorphanol sert tooltip serotonin transporter sris tooltip serotonin reuptake inhibitors selective serotonin reuptake inhibitors 6 nitroquipazine alaproclate bms 505130 centpropazine cericlamine citalopram dapoxetine desmethylcitalopram didesmethylcitalopram escitalopram femoxetine fluoxetine fluvoxamine indalpine ifoxetine madam norfluoxetine omiloxetine panuramine paroxetine pim 35 pirandamine rti 353 seproxetine sertraline zimelidine zinc000443438219 selective serotonin reuptake inhibitors and serotonin receptor modulators dsp 6745 etoperidone litoxetine lubazodone ly 393558 quipazine sb 649915 tgba01ad trazodone vilazodone vortioxetine serotonin norepinephrine reuptake inhibitors atomoxetine tomoxetine bicifadine cp 39332 desvenlafaxine duloxetine eclanamine levomilnacipran mcn5652 milnacipran n methyl pppa pppa tofenacin venlafaxine serotonin norepinephrine dopamine reuptake inhibitors 3 3 diphenylcyclobutanamine amifitadine ansofaxine bicifadine brasofensine centanafadine cocaine dasotraline desmethylsertraline desmethylsibutramine bts 54354 diclofensine didesmethylsibutramine bts 54505 dov 102677 dov 216303 exp 561 fezolamine hdmp 28 hp 505 indatraline jnj 7925476 jz iv 10 lafadofensine liafensine mazindol naphyrone nefazodone nefopam ns 2359 perafensine prc200 pridefine pudafensine sep 228431 sep 228432 sibutramine tedatioxetine tesofensine threohydrobupropion tropanes e g cocaine tricyclic antidepressants amitriptyline cianopramine clomipramine cyanodothiepin desipramine dosulepin dothiepin doxepin imipramine lofepramine nortriptyline pipofezine protriptyline others a 80426 amoxapine antihistamines e g brompheniramine chlorphenamine dimenhydrinate diphenhydramine mepyramine pyrilamine pheniramine tripelennamine antipsychotics e g loxapine ziprasidone arylcyclohexylamines e g 3 meo pcp esketamine ketamine methoxetamine phencyclidine cyclobenzaprine delucemine dextromethorphan dextrorphan efavirenz hypidone medifoxamine mesembrine mifepristone min 117 wf 516 n me 5 ht opioids e g dextropropoxyphene methadone pethidine meperidine levorphanol tapentadol tramadol roxindole svn 015 vmats tooltip vesicular monoamine transporters amiodarone amphetamines e g amphetamine methamphetamine mdma app azik bietaserpine deserpidine deutetrabenazine dihydrotetrabenazine efavirenz gbr 12935 gz 793a ibogaine ketanserin lobeline methoxytetrabenazine reserpine rose bengal tetrabenazine valbenazine vanoxerine gbr 12909 others unsorted cendifensine dat enhancers luteolin dat modulators agonist like sori 9804 sori 20040 antagonist like sori 20041 see also receptor signaling modulators monoamine releasing agents adrenergics dopaminergics serotonergics monoamine metabolism modulators monoamine neurotoxins v t e muscarinic acetylcholine receptor modulators machrs tooltip muscarinic acetylcholine receptors agonists 77 lh 28 1 ac 42 ac 260 584 aceclidine acetylcholine af30 af150 s af267b alvameline aqra 741 arecoline bethanechol butyrylcholine carbachol cdd 0034 cdd 0078 cdd 0097 cdd 0098 cdd 0102 cevimeline choline cis dioxolane desmethylclozapine norclozapine ethoxysebacylcholine guvacoline gxv 813 ex a8078 itameline ly 593 039 l 689 660 ly 2 033 298 mcna343 methacholine milameline muscarine ngx 267 ocvimeline oxotremorine pd 151 832 pilocarpine rs86 sabcomeline sdz 210 086 sebacylcholine suberyldicholine talsaclidine tazomeline thiopilocarpine vedaclidine vu 0029767 vu 0090157 vu 0152099 vu 0152100 vu 0238429 way 132 983 xanomeline ym 796 positive allosteric modulators anavex 3 71 af710b antagonists 3 quinuclidinyl benzilate 4 damp aclidinium bromide formoterol abediterol af dx 250 af dx 384 ambutonium bromide anisodamine anisodine antihistamines first generation e g brompheniramine buclizine captodiame chlorphenamine chlorpheniramine cinnarizine clemastine cyproheptadine dimenhydrinate dimetindene diphenhydramine doxylamine meclizine mequitazine perlapine phenindamine pheniramine phenyltoloxamine promethazine propiomazine triprolidine aq ra 741 atropine atropine methonitrate atypical antipsychotics e g clozapine fluperlapine olanzapine fluoxetine rilapine quetiapine tenilapine zotepine benactyzine benzatropine benztropine benzilone benzilylcholine mustard benzydamine bevonium bibn 99 biperiden bornaprine camylofin car 226 086 car 301 060 car 302 196 car 302 282 car 302 368 car 302 537 car 302 668 caramiphen cimetropium bromide clidinium bromide cloperastine cs 27349 cyclobenzaprine cyclopentolate darifenacin dau 5884 desfesoterodine dexetimide dibd dicycloverine dicyclomine dihexyverine difemerine diphemanil metilsulfate ditran drofenine ea 3167 ea 3443 ea 3580 ea 3834 emepronium bromide etanautine etybenzatropine ethybenztropine fenpiverinium fentonium bromide fesoterodine flavoxate glycopyrronium bromide beclometasone formoterol indacaterol neostigmine hexahydrodifenidol hexahydrosiladifenidol hexbutinol hexocyclium himbacine hl 031 120 homatropine imidafenacin ipratropium bromide salbutamol isopropamide j 104 129 hyoscyamine mamba toxin 3 mamba toxin 7 mazaticol mebeverine meladrazine mepenzolate methantheline methoctramine methylatropine methylhomatropine methylscopolamine metixene muscarinic toxin 7 n ethyl 3 piperidyl benzilate n methyl 3 piperidyl benzilate nefopam octatropine methylbromide anisotropine methylbromide orphenadrine otenzepad af dx 116 otilonium bromide oxapium iodide oxitropium bromide oxybutynin oxyphencyclimine oxyphenonium bromide pbid pd 102 807 pd 0298029 penthienate pethidine pfhhsid phenglutarimide phenyltoloxamine pipenzolate bromide piperidolate pirenzepine piroheptine pizotifen poldine pridinol prifinium bromide procyclidine profenamine ethopropazine propantheline bromide propiverine quinidine 3 quinuclidinyl thiochromane 4 carboxylate revefenacin rociverine ru 47 213 sch 57 790 sch 72 788 sch 217 443 scopolamine hyoscine scopolamine butylbromide hyoscine butylbromide silahexacyclium sofpironium bromide solifenacin ssris tooltip selective serotonin reuptake inhibitors e g femoxetine paroxetine telenzepine terodiline tetracyclic antidepressants e g amoxapine maprotiline mianserin mirtazapine tiemonium iodide timepidium bromide tiotropium bromide tiquizium bromide tofenacin tolterodine tricyclic antidepressants e g amitriptyline perphenazine amitriptylinoxide butriptyline cidoxepin clomipramine desipramine desmethyldesipramine dibenzepin dosulepin dothiepin doxepin imipramine lofepramine nitroxazepine northiaden desmethyldosulepin nortriptyline protriptyline quinupramine trimipramine tridihexethyl trihexyphenidyl trimebutine tripitamine tripitramine tropacine tropatepine tropicamide tropine benzilate trospium chloride typical antipsychotics e g chlorpromazine chlorprothixene cyamemazine cyamepromazine loxapine mesoridazine thioridazine umeclidinium bromide vilanterol win 2299 xanomeline zamifenacin precursors and prodrugs acetyl coa adafenoxate choline lecithin citicoline cyprodenate dimethylethanolamine glycerophosphocholine meclofenoxate centrophenoxine phosphatidylcholine phosphatidylethanolamine phosphorylcholine pirisudanol see also receptor signaling modulators nicotinic acetylcholine receptor modulators acetylcholine metabolism transport modulators v t e nicotinic acetylcholine receptor modulators nachrs tooltip nicotinic acetylcholine receptors agonists and pams tooltip positive allosteric modulators 5 hiaa 6 chloronicotine a 84 543 a 366 833 a 582 941 a 867 744 abt 202 abt 418 abt 560 acetylcholine altinicline anabasine anatabine anatoxin a ar r17779 bephenium hydroxynaphthoate butinoline butyrylcholine carbachol choline choline m bromophenyl ether cotinine cytisine decamethonium desformylflustrabromine dianicline dimethylphenylpiperazinium epibatidine epiboxidine ethanol alcohol ethoxysebacylcholine evp 4473 evp 6124 galantamine gts 21 ispronicline ivermectin jnj 39393406 levamisole lobeline mem 63 908 rg 3487 morantel nicotine tobacco ns 1738 nndmai pha 543 613 pha 709 829 pnu 120 596 pnu 282 987 pozanicline pyrantel rivanicline rjr 2429 sazetidine a sb 206553 sebacylcholine sib 1508y sib 1553a sofinicline abt 894 ssr 180 711 suberyldicholine suxamethonium succinylcholine suxethonium succinyldicholine tc 1698 tc 1734 tc 1827 tc 2216 tc 5214 tc 5619 tc 6683 tebanicline tribendimidine tropisetron ub 165 varenicline way 317 538 xy 4083 antagonists and nams tooltip negative allosteric modulators 18 mac 18 mc α neurotoxins e g α bungarotoxin α cobratoxin α conotoxin many others abt 126 alcuronium allopregnanolone amantadine anatruxonium aqw051 atracurium barbiturates e g pentobarbital sodium thiopental bnc 210 bungarotoxins e g α bungarotoxin κ bungarotoxin bupropion bw284c51 bw a444 candocuronium iodide chandonium iodide chlorisondamine cisatracurium coclaurine coronaridine curare cyclopropane dacuronium bromide decamethonium dehydronorketamine desflurane dextromethorphan dextropropoxyphene dextrorphan diadonium dhβe dihydrochandonium dimethyltubocurarine metocurine dioscorine dipyrandium dizocilpine mk 801 doxacurium encenicline enflurane erythravine esketamine fazadinium gallamine gantacurium chloride halothane hexafluronium hexamethonium benzohexonium hydroxybupropion hydroxynorketamine ibogaine isoflurane ketamine kynurenic acid laudanosine laudexium laudolissin levacetylmethadol levomethadone malouetine me 18 mc mecamylamine memantine methadone methorphan racemethorphan methyllycaconitine metocurine mivacurium morphanol racemorphan neramexane nitrous oxide norketamine pancuronium bromide pempidine pentamine pentolinium phencyclidine pipecuronium bromide progesterone promegestone radafaxine rapacuronium bromide reboxetine rocuronium bromide sevoflurane stercuronium iodide surugatoxin thiocolchicoside threohydrobupropion toxiferine tramadol trimetaphan camsilate trimethaphan camsylate tropeinium tubocurarine vanoxerine vecuronium bromide xenon precursors and prodrugs acetyl coa adafenoxate choline lecithin citicoline cyprodenate dimethylethanolamine glycerophosphocholine meclofenoxate centrophenoxine phosphatidylcholine phosphatidylethanolamine phosphorylcholine pirisudanol see also receptor signaling modulators muscarinic acetylcholine receptor modulators acetylcholine metabolism transport modulators v t e opioid receptor modulators μ opioid mor agonists abridged full list 3 ho pcp 7 acetoxymitragynine 7 hydroxymitragynine ψ akuammigine α chlornaltrexamine α narcotine acetyldihydrocodeine acetylfentanyl acrylfentanyl adrenorphin metorphamide ah 7921 akuammicine akuammidine alfentanil anileridine apparicine β endorphin bam 12p bam 18p bam 22p benzhydrocodone benzylmorphine bezitramide biphalin bu08070 buprenorphine butorphan butorphanol butyrfentanyl bw373u86 carfentanil casokefamide cebranopadol chloroxymorphamine codeine dadle damgo dago dermorphin desmetramadol desmethyltramadol desomorphine deumitragynine dextromoramide dextropropoxyphene propoxyphene dezocine dimenoxadol dimethylaminopivalophenone eluxadoline diamorphine heroin dihydrocodeine dihydroetorphine dihydromorphine dinalbuphine sebacate diphenoxylate dipipanone dynorphin a embutramide endomorphin 1 endomorphin 2 eseroline ethylmorphine etorphine fentanyl fluorophen frakefamide furanylfentanyl hemorphin 4 herkinorin hodgkinsine hydrocodone hydromorphinol hydromorphone ibntxa ketamine ketobemidone kratom laudanosine lefetamine leu enkephalin levacetylmethadol levomethorphan levorphanol lexanopadol loperamide loxicodegol ls 115509 matrine meb 1170 meptazinol met enkephalin metenkefalin methadone metkefamide metopon mitragynine mitragynine pseudoindoxyl morphiceptin morphine nalbuphine naloxone benzoylhydrazone nalbzoh nalmexone naltalimide neopine nfepp nicocodeine nicodicodine nicomorphine norketamine nufenoxole octreotide oliceridine oxycodegol nktr 181 oxymorphone 3 methoxynaltrexonazine om 3 mnz oripavine oxycodone oxymorphazone oxymorphonazine oxymorphone oxymorphone phenylhydrazone oxypnph papaver somniferum opium pentazocine pericine pethidine meperidine phenazocine phencyclidine piminodine piritramide pl 017 prodine propiram pzm21 racemethorphan racemorphan remifentanil salsolinol sc 17599 sinomenine sr 15099 sr 17018 sufentanil susineridine tapentadol tetrahydropapaveroline th 030418 thebaine thienorphine tianeptine tilidine tramadol trimebutine trimu 5 trv734 tubotaiwine u 47700 valorphin viminol xorphanol antagonists 3s 4s picenadol 2 s n n r viminol 3cs nalmefene 4 caffeoyl 1 5 quinide 4 hydroxyflavanone 4 7 dihydroxyflavone 6β naltrexol 6β naltrexol d4 18 mc α gliadin β chlornaltrexamine β funaltrexamine akuammine alvimopan am 251 apigenin at 076 axelopran bevenopran catechin catechin gallate clocinnamox ctap ctop cyclofoxy cyprodime diacetylnalorphine diprenorphine ecg egc epicatechin eptazocine gemazocine ginsenoside r hyperoside ibogaine jdtic levallorphan lobeline ly 255582 ly 2196044 methocinnamox methylnaltrexone methylsamidorphan naldemedine nalmefene nalodeine n allylnorcodeine nalorphine nalorphine dinicotinate naloxazone naloxegol naloxol naloxonazine naloxone naltrexazone naltrexonazine naltrexone naltrindole naringenin noribogaine oxilorphan pawhuskin a rimonabant quadazocine samidorphan taxifolin δ opioid dor agonists 3cs nalmefene 6 gnti 7 siom adl 5747 pf 04856881 adl 5859 alazocine skf 10047 amoxapine ar m100390 arm390 azd2327 β endorphin bam 18p biphalin bu 48 butorphan butorphanol bw373u86 casokefamide cebranopadol codeine cyclazocine dadle deltorphin a deltorphin i deltorphin ii desmethylclozapine desmetramadol desmethyltramadol dezocine diamorphine heroin dihydroetorphine dihydromorphine dpdpe dpi 221 dpi 3290 dslet ethylketazocine etorphine fentanyl fit fluorophen hemorphin 4 hydrocodone hydromorphone ibogaine isomethadone jnj 20788560 knt 127 kratom laudanosine leu enkephalin levomethorphan levorphanol lexanopadol lofentanil met enkephalin metenkefalin metazocine metkefamide mitragynine mitragynine pseudoindoxyl morphine n phenethyl 14 ethoxymetopon norbuprenorphine nalbzoh oripavine oxycodone oxymorphone pethidine meperidine proglumide racemethorphan racemorphan rwj 394674 samidorphan sb 235863 snc 80 snc 162 tan 67 sb 205 607 th 030418 thebaine thiobromadol c 8813 tonazocine tramadol trv250 xorphanol zenazocine antagonists 4 7 dihydroxyflavone 5 ntii 6β naltrexol 6β naltrexol d4 α santolol β chlornaltrexamine apigenin at 076 axelopran bevenopran bntx catechin catechin gallate clocinnamox diacetylnalorphine...
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